Publikacje

Cytotoxic effects of halophilic archaea metabolites on ovarian cancer cell lines
Kowalewicz-Kulbat, K. T. Krawczyk, I. Szulc-Kiełbik, S. Rykowski, M. Denel-Bobrowska, A. B. Olejniczak, C. Locht, M. Klink
Microb. Cell. Fact. 2023, 22, 197, doi/org/10.1186/s12934-023-02206-y

Synthesis and in vitro cytotoxic activity of dye-linker-macrocycle conjugates with variable linker length and components
M. D. Tomczyk, K. Matczak, M. Skonieczna, P. Chulkin, M. Denel-Bobrowska, D. Różycka, S. Rykowski, A. B. Olejniczak, K. Walczak
Bioorg. Chem. 2023, 140, 106782, doi.org/10.1016/j.bioorg.2023.106782

Acridine/acridone-carborane conjugates as strong DNA-binding agents with anticancer potential
D. Różycka, A. Kowalczyk, M. Denel-Bobrowska, O. Kuźmycz, M. Gapińska, P. Stączek, A. B. Olejniczak
ChemMedChem 2023, e202200666, doi: 10.1002/cmdc.202200666

Carboranyl-1,8-naphthalimide intercalators indice lysosomal membrane permeabilization and ferroptosis in cancer cell line
S. Rykowski, D. Gurda-Woźna, A. Fedoruk-Wyszomirska, M. Orlicka-Płocka, Aleksandra Kowalczyk, P. Stączek, M. Denel-Bobrowska, A. Biniek-Antosiak, W. Rypniewski, E. wyszko, A. B. Olejniczak
J. Enzym. Inhib. Med. Chem. 2023, 38(1), 2171028, doi: 10.1080/14756366.2023.2171028

Chiral 2-azabicycloalkanes bearing 1,2,3-triazole, thiourea, and ebselen moieties – synthesis and biological activity
F. Steppeler, D. Iwan, R. Gaida, M. Denel-Bobrowska, A. B. Olejniczak, E. Wojaczyńska
Biomed. Pharmacother. 2023, 164, 114908, doi: 10.1016/j.biopha.2023.114908

Non-nucleoside structured compound with antiviral activity – past 10 years (2010-2020)
M. Denel-Bobrowska, A. B. Olejniczak
Eur. J. Med. Chem. 2022, 231, 114136, doi: 10.1016/j.ejmech.2022.114136

Nematicidal activity of naphthalimide-boron cluster conjugates
A.Bogucka-Kocka, P. Kołodziej, A. Makuch-Kocka, D. Różycka, S. Rykowski, J. Nekvinda, B. Gruner, A. B. Olejniczak
Chem. Commun. 2022, 58, 2528-2531, doi: 10.1039/d1cc07075d

Design of DNA intercalators based on 4-carboranyl-1,8-naphthalimides: investigation of their DNA-binding ability and anticancer activity,
S. Rykowski, D. Gurda-Woźna, M. Orlicka-Płocka, A. Fedoruk-Wyszomirska, M. Giel-Pietraszuk, E. Wyszko, A. Kowalczyk, P. Stączek, K. Biniek-Antosiak, W. Rypniewski, A. B. Olejniczak
Int. J. Mol. Sci. 2022, 23, 4598, doi: 10.3390/ijms23094598

Fluorinated analogues of lepidilines A and C: synthesis and screening of their anticancer and antiviral activity
G. Mloston, M. Kowalczyk, M. Celeda, M. Jasiński, M. Denel-Bobrowska, A. B. Olejniczak
Molecules 2022, 27, 3524, doi: 10.3390/molecules27113524

Chiral sulfonamides with various N-heterocyclic and aromatic units – synthesis and antiviral activity evaluation
D. Iwan, K. Kamińska, M. Denel-Bobrowska, A. B. Olejniczak, E. Wojaczyńska
Biomed. Pharmacother. 2022, 153, 113473, doi: 10.1016/j.biopha.2022.113473

Design, synthesis, and evaluation of novel 3-carboranyl-1,8-naphthalimide derivatives as potential anticancer agents
S. Rykowski, D. Gurda-Woźna, M. Orlicka-Płocka, A. Fedoruk-Wyszomirska, M. Giel-Pietraszuk, E. Wyszko, A. Kowalczyk, P. Stączek, A. Bąk, A. Kiliszek, W. Rypniewski, A. B. Olejniczak,
Int. J. Mol. Sci. 2021, 22(5), 2772, doi: 10.3390/ijms22052772

In vitro anticancer and antivirus activities of cyano- and bis(trifluorometylsulfonyl)imide-based ionic liquids
M. Musiał, A. B. Olejniczak, M. Denel-Bobrowska, E. Zorębski, M. Dzida
ACS Sustain. Chem. Eng. 2021, 9. 16459-16465, doi: 10.1021/acssuschemeng.1c06580

Synthesis of naphthalimide-carborane and metallacarborane conjugates: anticancer activity, DNA binding ability
J. Nekvinda, D. Różycka, S. Rykowski, E. Wyszko, A. Fedoruk-Wyszomirska, D. Gurda, M. Orlicka-Płocka, M. Giel-Pietraszuk, A. Kiliszek, W. Rypniewski, R. Bachorz, J. Wojcieszak, B. Gruner, A. B. Olejniczak
Bioorganic Chem. 2020, 94, 103432, doi: 10.1016/j.bioorg.2019.103432

Novel isoniazid-carborane hybrids active in vitro against Mycobacterium tuberculosis, D. Różycka, M. Korycka-Machała, A. Żaczek, J. Dziadek, D. Gurda, M. Orlicka-Płocka, E. Wyszko, K. Biniek-Antosiak, W. Rypniewski, A. B. Olejniczak,
Pharmaceuticals, 2020, 13, 465, doi:10.3390/ph13120465.

Comparative DFT study of inclusion complexes of thymin-carborane conjugate with ß-cyclodextrin and heptakis (2,6-O-dimethyl)-ß-cyclodextrin in water
A.Ignaczak, Ł. Orszański, M. Adamiak, A. B. Olejniczak
J. Mol. Liq. 2020, 315, 113767, doi: 10.1016/j.molliq.2020.113767

(1-4)-Thiodisaccharides as anticancer agnts. Part 5. Evaluation of anticancer activity and investigation of mechanism of action
J. Sarnik, A. Gajek, M. Toma, J. Pawelczyk, S. Rykowski, A. Olejniczak, T. Sliwinski, R. Bielski, Z. J. Witczak
Bioorg. Med. Chem. Lett. 2020, 30, 126904, doi: 10.1016/j.bmcl.2019.126904

PPE51 is involved in the uptake of disaccharides by Mycobacterium tuberculosis
M. Korycka-Machała, J. Pawełczyk, P. Borówka, B. Dziadek, A. Brzostek, M. Kawka, A. Bekier, S. Rykowski, A. B. Olejniczak, S. Strapagiel, Z. Witczak, J. Dziadek,
Cells, 2020, 9, 603, doi:10.3390/cells9030603